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CAPROOYL TETRAPEPTIDE-3 AMIDE.

Valuable / SKIN CONDITIONING

An advanced, biomimetic signaling molecule designed to replicate the activity of natural protease inhibitors to reinforce skin architecture. This specific amide-modified version offers superior enzymatic stability, making it a high-performance choice for restructuring the dermal-epidermal junction.

Cell-Communicating Ingredient Skin Conditioning Anti-Aging Structural Reinforcement

Science

This peptide functions by mimicking the activity of Elafin, a natural protease inhibitor. It communicates directly with skin cells to stimulate the synthesis of essential structural proteins, specifically Laminin-5, Collagen VII, and Fibronectin, which serve as the 'glue' for the Dermal-Epidermal Junction (DEJ) to ensure skin firmness and cohesion.


Research

High confidence
Effective range 1–2.5%
Optimal

2.5%

Key findings

  1. 01 A 28-day clinical evaluation of the base peptide at 2.5% demonstrated a reduction in fine line and wrinkle depth by up to 29% through DEJ reinforcement.
  2. 02 Independent clinical testing on proprietary peptide blends containing this ingredient showed measurable improvements in barrier function, hydration, and skin texture within 4 weeks of consistent application.

Transparency

Commonly dusted
Min. effective
1%
Red flag below
0.5%

Due to its high cost and efficacy at low levels, many mass-market products include this peptide at 'claim' levels (under 0.5%). For meaningful structural improvement and a reduction in wrinkle depth, concentrations should ideally align with the 2.5% clinical benchmark.


The Formula

Solubility
Water
Optimal pH 4.5 – 7
0 7 14

Stability

The C-terminus amide modification provides enhanced resistance against degradation by proteolytic enzymes. It is thermo-sensitive and must be incorporated during the cooling phase of production (below 40°C).

Synergies

  • Hyaluronic acid
  • Niacinamide
  • Non-acidic antioxidants

Conflicts

  • Strong oxidizing agents
  • AHA/BHA formulations below pH 4.0
  • Proteolytic enzymes (Papain, Bromelain)

Safety

CIR Status
Safe as used
Max tested
2.5%
Pregnancy
Safe
Sensitization risk Low

Classified as safe for cosmetic use with a low risk profile; it is non-sensitizing and generally well-tolerated by reactive skin types.


Your Skin

Yes Normal
Yes Dry
Yes Oily
Yes Sensitive
Irritancy Low
Comedogenicity Low

Our Assessment

Valuable

A precise, evidence-based peptide that delivers significant structural improvement and wrinkle reduction when formulated at clinical concentrations.


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References