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CAFFEOYL HEXAPEPTIDE-43.

Valuable / ANTIOXIDANT, SKIN PROTECTING

A cutting-edge peptide-drug conjugate (PDC) that molecularly bridges caffeic acid with a silkworm-derived hexapeptide for enhanced stability and biological activity. This bio-engineered molecule provides a robust shield against oxidative stress while simultaneously calming inflammatory pathways within the skin matrix.

Antioxidant Anti-inflammatory Skin-protecting DNA-protection

Science

This ingredient functions as a high-affinity antioxidant by neutralizing DPPH, hydroxyl, and peroxyl radicals. By linking caffeic acid to the APPPKK peptide sequence, it achieves superior cellular delivery, where it inhibits the production of nitric oxide (NO) to reduce inflammation and prevents DNA damage and lipid peroxidation caused by hydrogen peroxide exposure.


Research

Medium confidence
Effective range 0.001–0.01%
Optimal

0.007%

Key findings

  1. 01 In vitro analysis (Lee et al., 2017) demonstrated that at a 100 μM concentration (0.007%), the peptide achieved 87.3% radical scavenging activity and significant suppression of inflammatory markers while maintaining over 90% cell viability.

Transparency

Commonly dusted
Min. effective
0.005%
Red flag below
0.001%

Because this peptide is bioactive at extremely low concentrations (parts per million), many formulations include it at 'label-only' levels. For meaningful antioxidant protection, it should be present at or near the 0.007% (70 ppm) concentration used in primary research.


The Formula

Solubility
Water
Optimal pH 5 – 7
0 7 14

Stability

The conjugation process significantly improves the water solubility and oxidative stability of caffeic acid, preventing the common browning and degradation often seen with free phenolic acids.

Synergies

  • Vitamin C
  • Hyaluronic acid
  • Niacinamide

Conflicts

  • Strong oxidizing agents
  • Strong acids
  • Strong bases
  • Proteolytic enzymes

Safety

CIR Status
Not reviewed
Pregnancy
Safe
Sensitization risk Low

As a relatively recent biotech innovation, it lacks a formal CIR review, but initial toxicological data shows high cell viability and low irritation potential.


Your Skin

Yes Normal
Yes Dry
Yes Oily
Yes Sensitive
Irritancy Low
Comedogenicity Low

Our Assessment

Valuable

A sophisticated, high-stability antioxidant peptide that offers precise protection against environmental DNA damage and inflammation.


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