Get a Free 5ml Mini Now Free 5ml Mini With Every Order of The Mantle

TOCOPHERYL DIMETHYLGLYCINATE.

Valuable CAS 124508-70-9 / ANTIOXIDANT, SKIN CONDITIONING

Tocopheryl Dimethylglycinate is a sophisticated, water-soluble derivative of gamma-tocopherol, engineered as a prodrug to deliver targeted antioxidant protection and contribute to effective skin lightening within the dermal layers.

Antioxidant Skin Conditioning Skin Lightening

Science

Upon topical application, Tocopheryl Dimethylglycinate undergoes enzymatic conversion within the skin to its active form, gamma-tocopherol (gamma-Toc). This potent antioxidant then effectively neutralizes free radicals, mitigating oxidative stress and cellular damage. Furthermore, gamma-Toc directly intervenes in the melanin synthesis pathway, leading to a visible reduction in pigmentation.


Research

Medium confidence
Effective range 0.1–0.5%
Optimal

0.5%

Key findings

  1. 01 A 0.5% topical application demonstrated significant skin lightening, reducing pigmentation by 70% in UVB/UVA-exposed brownish guinea pigs compared to irradiated controls.
  2. 02 In vitro studies utilizing murine B16 melanoma cells showed that gamma-TDMG, at concentrations of 0.1% or 0.5%, effectively suppressed melanin synthesis.

Transparency

Not commonly dusted

The Formula

Solubility
Water
Optimal pH N/A
0 7 14

Stability

Identified as a hydrophilic and water-soluble derivative of gamma-tocopherol, suggesting enhanced stability compared to free tocopherol in aqueous environments. This water-soluble nature makes it a stable vitamin E prodrug for aqueous formulations.


Safety

CIR Status
Not reviewed
Sensitization risk Unknown

While commonly used as a cosmetic antioxidant and skin conditioning agent, Tocopheryl Dimethylglycinate lacks specific safety assessments from major regulatory bodies such as CIR, SCCS, or FDA as a distinct ingredient. Its safety profile is generally inferred from the well-established safety of general tocopherols, though ingredient-specific comprehensive data remains to be publicly detailed.


Your Skin

No Normal
No Dry
No Oily
No Sensitive
Irritancy Unknown
Comedogenicity Unknown

Our Assessment

Valuable

Tocopheryl Dimethylglycinate is a valuable water-soluble Vitamin E derivative offering significant antioxidant protection and promising skin lightening capabilities through melanin inhibition.


Related

Finding similar ingredients…